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المعرفة
بحث
قالب
:
Glutamate receptor ligands
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عدل
v
t
e
Glutamate receptor
ligands
Ionotropic
NMDA
Agonists
;
NMDA
•
Tetrazolylglycine
Antagonists
;
Competitive antagonists
;
AP7
•
AP5
•
CGP-37849
•
Midafotel (CPPene)
•
PEAQX
•
Perzinfotel
•
PPDA
•
Sdz 220-581
•
Selfotel
;
Noncompetitive antagonists
;
Aptiganel
•
Dizocilpine
•
FPL-12495
•
FR-115,427
•
Gacyclidine
•
Hodgkinsine
•
HU-211
•
Indantadol
•
Psychotridine
•
Remacemide
;
Uncompetitive channel blockers
;
2-MDP
•
8a-Phenyldecahydroquinoline
•
Amantadine
•
Budipine
•
Delucemine
•
Dexoxadrol
•
Dextromethorphan
•
Dextrorphan
•
Endopsychosin
•
Etoxadrol
•
Eticyclidine
•
Ibogaine
•
كتامين
•
Memantine
•
NEFA
•
Neramexane
•
Nitrous oxide
•
Phencyclidine
•
Rhynchophylline
•
Riluzole
•
Rolicyclidine
•
Tenocyclidine
•
Tiletamine
•
Xenon
;
Glycine site antagonists
;
1-Aminocyclopropanecarboxylic acid
•
ACEA-1021
•
7-Chlorokynurenate
•
CGP-39653
•
DCKA
•
Gavestinel
•
GV-150,526
•
Kynurenic acid
•
L-689,560
•
Lacosamide
•
ZD-9379
;
Polyamine site antagonists
;
Besonprodil
•
CP-101,606
•
Eliprodil
•
Ifenprodil
•
Ro25-6981
•
Traxoprodil
;
Indirect antagonists
;
Lubeluzole
AMPA
Agonists
;
AMPA
•
Domoic acid
•
5-Fluorowillardiine
;
Positive allosteric modulators
;
Aniracetam
•
Cyclothiazide
•
CX-516
•
CX-546
•
CX-614
•
CX-691
•
CX-717
•
IDRA-21
•
LY-392,098
•
LY-404,187
•
LY-451,395
•
LY-451,646
•
LY-503,430
•
Oxiracetam
•
PEPA
•
Piracetam
•
Pramiracetam
Antagonists
;
ATPO
•
CNQX
•
DNQX
•
NBQX
•
Tezampanel (LY-293,558)
;
Negative allosteric modulators
;
GYKI-53,655
Kainate
Agonists
;
5-Iodowillardiine
•
ATPA
•
Domoic acid
•
Kainic acid
•
LY-339,434
•
SYM-2081
Antagonists
;
CNQX
•
DNQX
•
LY-382,884
•
NBQX
•
NS102
•
UBP-302
;
Negative allosteric modulators
;
NS-3763
Metabotropic
Group I
Agonists
;
Unselective
;
ACPD
•
Dihydroxyphenylglycine
;
mGlu1 selective
;
Ro01-6128
;
mGlu5 selective
;
CHPG
•
DFB
Antagonists
;
Unselective
;
MCPG
;
mGlu1 selective
;
BAY 36-7620
•
CPCCOEt
•
LY-367,385
;
mGlu5 selective
;
LY-344,545
•
MPEP
•
MTEP
Group II
Agonists
;
Unselective
;
Eglumegad (LY-354,740)
•
LY-404,039
;
mGlu2 selective
;
BINA
•
LY-487,379
Antagonists
;
EGLU
•
LY-341,495
Group III
Agonists
;
Unselective
;
AP4
;
mGlu4 selective
;
PHCCC
;
mGlu8 selective
;
DCPG
Antagonists
;
CPPG
•
UBP-1112